Prof. Dr. Peter Gmeiner

Lehrstuhl für Pharmazeutische Chemie

Interactive SAR Studies: Rational Discovery of Super-Potent and Highly Selective Dopamine D3 Receptor Antagonists and Partial Agonists (2002) Gmeiner P, Hübner H Journal article Fused Azaindole Derivatives: Molecular Design, Synthesis and in vitro Pharmacology Leading to the Preferential Dopamine D3 Receptor Agonist FAUC 725 (2002) Löber S, Gmeiner P, Hübner H Journal article Di- and Trisubstituted Pyrazolo[1,5-a]pyridine Derivatives: Synthesis, Dopamine Receptor Binding and Ligand Efficacy (2002) Löber S, Gmeiner P, Hübner H Journal article Analogs of the dopamine D4 receptor ligand FAUC 113 with planar- and central-chirality (2002) Löber S, Gmeiner P, Hübner H Journal article 2,4-Disubstituted Pyrroles: Synthesis, Traceless Linking and Pharmacological Investigations Leading to the Dopamine D4 Receptor Partial Agonist FAUC 356 (2002) Gmeiner P, Hübner H Journal article Short and Efficient Synthesis of Homo-Freidinger Lactams: An Olefin Metathesis Approach Towards Conformationally Restricted ß-Amino Acid Analogues (2002) Gmeiner P Journal article Comparative molecular field analysis of dopamine D4 receptor antagonists including 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo-[2,3-b]pyridine (L-745,870), and clozapine. (2001) Lanig H, Utz W, Gmeiner P Journal article, Original article Comparative Molecular Field Analysis of Dopamine D4 Receptor Antagonists Including 3-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine (L-745,870), and Clozapine (2001) Lanig H, Utz W, Gmeiner P, Lanig H Journal article, Original article Synthesis and in vitro Evaluation of Iodine Labelled Pyrazolo[1,5-a]pyridines as Highly Selective Dopamine D4 Receptor Ligands (2001) Löber S, Gmeiner P, Hübner H Journal article Rationally Based Efficacy Tuning of Selective Dopamine D4 Receptor Ligands Leading to the Complete Antagonist 2-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213) (2001) Utz W, Löber S, Gmeiner P, Hübner H Journal article