Prof. Dr. Peter Gmeiner

Lehrstuhl für Pharmazeutische Chemie

Spontaneous butenolide ring formation of pregnane-21-O-malonyl hemiesters under mild reaction conditions is facilitated by the 14β-hydroxy group present in all natural cardenolides (2016) Maia de Pádua R, Meitinger N, Hennemann M, Schebitz P, Waibel R, Löber S, Gmeiner P, et al. Journal article, Original article Development of Covalent Ligand-Receptor Pairs to Study the Binding Properties of Nonpeptidic Neurotensin Receptor 1 Antagonists. (2016) Kling R, Plomer M, Lang C, Banerjee A, Hübner H, Gmeiner P Journal article, Original article Mimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples. (2016) Keller M, Kuhn KK, Einsiedel J, Hübner H, Biselli S, Mollereau C, Wifling D, et al. Journal article, Original article Comparative MD Simulations Indicate a Dual Role for Arg132(3.50) in Dopamine-Dependent D2R Activation (2016) Kling R, Clark T, Gmeiner P Journal article, Original article Structure-guided development of heterodimer-selective GPCR ligands (2016) Hübner H, Schellhorn T, Gienger M, Schaab C, Kaindl J, Leeb L, Clark T, et al. Journal article, Original article Optimization and synthesis of an 18F-labeled dopamine D3 receptor ligand using [18F]fluorophenylazocarboxylic tert-butylester (2016) Nebel N, Maschauer S, Hocke C, Hübner H, Gmeiner P, Prante O Journal article, Original article 18F- and 68Ga-Labeled Neurotensin Peptides for PET Imaging of Neurotensin Receptor 1 (2016) Maschauer S, Einsiedel J, Hübner H, Gmeiner P, Prante O Journal article, Original article The broad-spectrum antiinfective drug artesunate interferes with the canonical nuclear factor kappa B (NF-κB) pathway by targeting RelA/p65 (2015) Hutterer C, Niemann I, Milbradt J, Fröhlich T, Reiter C, Kadioglu O, Bahsi H, et al. Journal article, Original article Multicomponent Synthesis and Biological Evaluation of a Piperazine-Based Dopamine Receptor Ligand Library (2015) Stucchi M, Gmeiner P, Hübner H, Rainoldi G, Sacchetti A, Silvani A, Lesma G Journal article, Original article Covalent molecular probes for class A G protein-coupled receptors: advances and applications (2015) Weichert D, Gmeiner P Journal article, Review article