Lehrstuhl für Pharmazeutische Chemie

Synthesis, biological evaluation and radiolabelling by 18F- fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET (2010) Höfling S, Maschauer S, Hübner H, Gmeiner P, Wester HJ, Prante O, Heinrich M Journal article, Original article Functional characterization of a partial loss-of-function mutation of the epithelial sodium channel (ENaC) associated with atypical cystic fibrosis (2010) Huber R, Krüger B, Diakov A, Korbmacher J, Härteis S, Einsiedel J, Gmeiner P, et al. Journal article, Original article Engineering a GPCR-ligand pair that simulates the activation of D 2L by dopamine (2010) Tschammer N, Doerfler M, Hübner H, Gmeiner P Journal article, Original article Click-chemistry-derived tetracycline-amino acid conjugates exhibiting exceptional potency and exclusive recognition of the reverse tet repressor (2010) Usai I, Krüger M, Einsiedel J, Hillen W, Gmeiner P Journal article, Original article Anhydrotetracycline-peptide conjugates as representatives for ligand-based transactivating systems (2010) Lochner S, Einsiedel J, Schaefer G, Berens C, Hillen W, Gmeiner P Journal article, Original article Bioisosteric replacement leading to biologically active [2.2]Paracyclophanes with altered binding profiles for aminergic g-protein-coupled receptors (2010) Skultety M, Hübner H, Löber S, Gmeiner P Journal article, Original article Labeling and glycosylate of peptides using click chemistry: a general approach to18F-glycopeptides as effective imaging probes for positron emission tomography (2010) Maschauer S, Einsiedel J, Haubner R, Hocke C, Ocker M, Hübner H, Kuwert T, et al. Journal article A series of 18F-labelled pyridinylphenyl amides as subtype-selective radioligands for the dopamine D3 receptor (2010) Hocke C, Maschauer S, Hübner H, Löber S, Utz W, Kuwert T, Gmeiner P, Prante O Journal article Quinpramine is a novel compound effective in ameliorating brain autoimmune disease (2009) Singh MP, Hoerste GMZ, Hu W, Mausberg AK, Cravens PD, Eagar T, Löber S, et al. Journal article Parallel synthesis of potent dopaminergic N-phenyltriazole carboxamides applying a novel click chemistry based phenol linker (2009) Loaiza PR, Löber S, Hübner H, Gmeiner P Journal article, Original article