Lehrstuhl für Pharmazeutische Chemie

The bulky N(6) substituent of cabergoline is responsible for agonism of this drug at 5-hydroxytryptamine (5-HT)2A and 5-HT2B receptors and thus is a determinant of valvular heart disease (2011) Kekewska A, Hübner H, Gmeiner P, Pertz HH Journal article, Original article Histidine 6.55 is a major determinant of ligand-biased signaling in dopamine D2L receptor (2011) Tschammer N, Bollinger S, Kenakin T, Gmeiner P Journal article, Original article Aromatic ring functionalization of benzolactam derivatives: New potent dopamine D3 receptor ligands (2011) Ortega R, Hübner H, Gmeiner P, Masaguer CF Journal article, Original article A highly efficient type I β-turn mimetic simulating an asx-pro-turn-like structure (2011) Pinsker A, Einsiedel J, Härterich S, Waibel R, Gmeiner P Journal article, Original article Structural Basis for Species Selectivity in the HIV-1 gp120-CD4 Interaction: Restoring Affinity to gp120 in Murine CD4 Mimetic Peptides (2011) Kaßler K, Meier J, Eichler J, Sticht H Journal article Novel pyridylmethylamines as highly selective 5-HT1A superagonists (2010) Bollinger S, Hübner H, Heinemann FW, Meyer K, Gmeiner P Journal article, Original article 4-substituted tert-butyl phenylazocarboxylates-synthetic equivalents for the para-phenyl radical cation (2010) Höfling S, Bartuschat A, Heinrich M Journal article, Original article The therapeutically anti-prion active antibody-fragment scF v-W226: Paramagnetic relaxation-enhanced NMR spectroscopy aided structure elucidation of the paratope-epitope interface (2010) Mangels C, Kellner R, Einsiedel J, Weiglmeier PR, Rösch P, Gmeiner P, Schwarzinger S Journal article, Original article Tetracycline sensing using novel doxycycline derivatives immobilized on different surface plasmon resonance biosensor surfaces (2010) Andree U, Müller-Seitz E, Usai I, Löber S, Gmeiner P, Wimmer C, Hillen W, Petz M Journal article, Original article Synthesis of a 68Ga-labeled peptoid?peptide hybrid for imaging of neurotensin receptor expression in vivo (2010) Maschauer S, Einsiedel J, Hocke C, Hübner H, Kuwert T, Gmeiner P, Prante O Journal article, Original article