Journal of Medicinal Chemistry
Journal Abbreviation: J MED CHEM
ISSN: 0022-2623
eISSN: 1520-4804
Publisher: American Chemical Society
Publications (71)
Fancy Bioisosteres: Metallocene-Derived G-Protein-Coupled Receptor Ligands with Subnanomolar Binding Affinity and Novel Selectivity Profiles (2005)
Gmeiner P, Hübner H
Journal article
CoMFA and CoMSIA Investigations Revealing Novel Insights into the Binding Modes of Dopamine D3 Receptor Agonists (2005)
Hübner H, Gmeiner P, Utz W
Journal article
Evaluation of Lactam Bridged Neurotensin Analogues Adjusting psi(Pro10) Close to the Experimentally Derived Bioactive Conformation of NT(8-13) (2004)
Gmeiner P, Einsiedel J, Hübner H
Journal article
Systematic surface scan of the most favorable interaction sites of magnesium ions with tetracycline (2003)
Othersen O, Lanig H, Clark T
Journal article
Descriptors, physical properties, and drug-likeness (2002)
Brüstle M, Beck B, Schindler T, King W, Clark T
Journal article
Interactive SAR Studies: Rational Discovery of Super-Potent and Highly Selective Dopamine D3 Receptor Antagonists and Partial Agonists (2002)
Gmeiner P, Hübner H
Journal article
Comparative molecular field analysis of dopamine D4 receptor antagonists including 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo-[2,3-b]pyridine (L-745,870), and clozapine. (2001)
Lanig H, Utz W, Gmeiner P
Journal article, Original article
Comparative Molecular Field Analysis of Dopamine D4 Receptor Antagonists Including 3-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine (L-745,870), and Clozapine (2001)
Lanig H, Utz W, Gmeiner P, Lanig H
Journal article, Original article
Rationally Based Efficacy Tuning of Selective Dopamine D4 Receptor Ligands Leading to the Complete Antagonist 2-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213) (2001)
Utz W, Löber S, Gmeiner P, Hübner H
Journal article
Cyanoindole Derivatives as Highly Selective Dopamine D4 Receptor Partial Agonists: Solid-Phase Synthesis, Binding Assays, and Functional Experiments (2000)
Gmeiner P, Hübner H
Journal article