Journal of Medicinal Chemistry
Journal Abbreviation: J MED CHEM
ISSN: 0022-2623
eISSN: 1520-4804
Publisher: American Chemical Society
Publications (71)
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model (2008)
Kornhuber J, Tripal P, Reichel M, Terfloth L, Bleich S, Wiftfang J, Gulbins E
Journal article
Novel D3 Selective Dopaminergics Incorporating Enyne Units as Nonaromatic Catechol Bioisosteres: Synthesis, Bioactivity, and Mutagenesis Studies (2008)
Doerfler M, Tschammer N, Hamperl K, Hübner H, Gmeiner P
Journal article
Synthesis, Radiofluorination and In Vitro Evaluation of Pyrazolo[1,5-a]pyridine Based Dopamine D4 Receptor Ligands: Discovery of an Inverse Agonist Radioligand for PET (2008)
Prante O, Tietze R, Hocke C, Löber S, Hübner H, Kuwert T, Gmeiner P
Journal article
Structure-Selectivity Investigations of D2-like Receptor Ligands by CoMFA and CoMSIA Guiding the Discovery of D3 Selective PET Radioligands (2007)
Utz W, Prante O, Hübner H, Kuwert T, Gmeiner P
Journal article
Structural changes and binding characteristics of the tetracycline-repressor binding site on induction (2006)
Lanig H, Othersen O, Seidel U, Beierlein F, Exner T, Clark T
Journal article
Fancy Bioisosteres: Novel Paracyclophane Derivatives as Super-Affinity Dopamine D3 Receptor Antagonists (2006)
Gmeiner P, Hübner H
Journal article
A Chimeric Ligand Approach Leading to Potent Antiprion Active Acridine Derivatives: Design, Synthesis and Biological Investigations (2006)
Löber S, Gmeiner P
Journal article
2-[(4-Phenylpiperazin-1-yl)methyl]imidazo(di)azines as Selective D4-Ligands. Induction of Penile Erection by 2-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a Potent and Selective D4 Partial Agonist (2006)
Gmeiner P, Hübner H
Journal article
Pharmacophore-guided drug discovery investigations leading to bioactive 5-aminotetrahydropyrazolopyridines. Implications for the binding mode of heterocyclic dopamine D3 receptor agonists. (2005)
Gmeiner P, Heinemann FW
Journal article
Modeling the Similarity and Divergence of Dopamine D2-like Receptors and Identification of Validated Ligand-Receptor Complexes (2005)
Böckler F, Lanig H, Gmeiner P
Journal article, Original article